Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as

Nov 22, 2017 - Elena Sandoval, María José Lafuente-Monasterio, María J. Almela, Pablo ... Santiago Ferrer-Bazaga, María Teresa Fraile, Francisco J. Ga...
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Correction to The Discovery of Novel Antimalarial Aminoxadiazoles as a Promising Nonendoperoxide Scaffold Elena Sandoval, María José Lafuente-Monasterio, María J. Almela, Pablo Castañeda, María Belén Jiménez Díaz, María S. Martínez-Martínez, Jaume Vidal, Iń ̃igo Angulo-Barturen, Paul Bamborough, Jeremy Burrows, Nicholas Cammack, María J. Chaparro, José M. Coterón, Cristina de Cozar, Benigno Crespo, Beatriz Díaz, Gerard Drewes, Esther Fernández, Santiago Ferrer-Bazaga, María Teresa Fraile, Francisco J. Gamo, Sonja Ghidelli-Disse, Rubén Gómez, John Haselden, Sophie Huss, María Luisa León, Jaime de Mercado, Simon J. F. Macdonald, José Ignacio Martín Hernando, Sara Prats, Margarita Puente, Anne Rodríguez, Juan C. de la Rosa, Lourdes Rueda, Carolyn Selenski, Paul Willis, David M. Wilson, Michael Witty, and Félix Calderón* Journal of Medicinal Chemistry 2017, 60, 6880−6896. DOI: 10.1021/acs.jmedchem.6b01441 Page 6882. In step 2 of Scheme 1, route A, the reagent is incorrect. Carboxamide bearing an R1 group should be the corresponding hydrazide derivative as shown below. The experimental procedure is correct. Scheme 1. (corrected route A)

Published: November 22, 2017 © 2017 American Chemical Society

9911

DOI: 10.1021/acs.jmedchem.7b01491 J. Med. Chem. 2017, 60, 9911−9911