Irreversible enzyme inhibitors. CLXV. Proteolytic enzymes. 15

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C(SH,)=XH. HCI C(NHs)=SH, HCI C(NH?)=XH .2TsOH C (SH,)=NH TsOH C(X H?)=XH, HCl C(NH?)=KH. TsOH C(SH?)=NH .HC1 C(XH?)=NH.TYOH C (NH*)=SH ,2HC1 C(PU"2j=SH.Pirrate C (XH?)=N H , TsOH C(?;H2)=NH HCI C(NHI)=NH. HC1 C(NH?j=XH , ~ T s O H C(XH,)=NH .HC1 C(SH2 )=SH ,TsOH C (YHz)=SH HC1 C(XH?)=SH TsOH C (N HZ)=K H .TYOH C(SH2)=NH ,TsOH C(NH%)=NH,TsOH C(XH,)=KH .T+OH C(NHnj=?rTH, TsOH C(XH?)=XH TrOH C (YH?)=XH .Picrate C(NH,)=IU". Picrate C(KH?)=NH .TcOH CK CS CN ChT CY CN I

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94-9.i 146-1 49 191-192 12