Residential School on Medicinal Chemistry: R Biology and Chemistry of Drug Discovery June 3-7, 2013 Drew University, Madison, NJ The Residential School offers an intensive weeklong graduate-level course organized to provide an accelerated program for medicinal chemists, biologists and other industrial and academic scientists who wish to broaden their knowledge of drug discovery and development. The aim of the school is to concentrate on the fundamentals that are useful in drug discovery spanning initial target assay evaluation through clinical development. Several case histories of recent successful drug development programs will also be presented. The five-day program consists of lectures and case histories covering the following topics: Enzyme Inhibition Receptor Binding Assays Hit-to-Lead Process Fragment-based Drug Design Lead Discovery & Modification Structure-based Drug Design Drug-like Properties DMPK & Protein Binding
Molecular Modeling Chemoinformatics GPCRs Kinase Inhibitors Ion Channels Bioisosteres Preclinical Toxicology Clinical Development
William Greenlee, Vincent Gullo and Ronald Doll Co-organizers For more information and application forms: www.drew.edu/resmed e-mail:
[email protected] phone: 973/408-3787; fax: 973/408-3504
