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Author Index Ajani, J. Α., 31 Appendino, Giovanni, 262 Badham, Neil R, 326 Balasubramanian, S. V., I l l Bernacki, Ralph J., 262 Biediger, Ronald J., 288 Bignami, Gary, 81 Bissery, Marie-Christine, 262 Boatman, P. Douglas, 288 Boge, Thomas C , 217 Bourzat, J. D., 233 Bricard, L., 189 Campbell, S. J., 58 Carboni, J. M., 162 Casazza, A. M., 124 Caudle, Michael R., 173 Chen, Shu-Hui, 247 Chen, Thomas T., 173 Cheruvallath, Zacharia S., 217 Combeau, C , 262 Commerçon Α., 233 Conway, Simon P., 326 Croteau, Rodney, 72 Datta, Apurba, 217 Didier, Ε., 233 Dubois, J., 98,189 Duclos, Olivier, 262 Farina, Vittorio, 124,247 Fenoglio, Ivana, 262 Floreancig, Paul E., 326 Gaillard, C , 98 Gentile, Lisa N., 288 Georg, Gunda L, 217 Glass, Timothy E., 326 Grampovnik, D. J., 276 Grothaus, Paul, 81 Guénard, D., 189 Guéritte-Voegelein, F., 189 Guy, R. Κ., 302 Harriman, Géraldine C. B., 217
Hauck, S., 124 Heerding, Julie M., 154 Hefner, Jerry, 72 Hepperle, Michael, 217 Hezari, Mehri, 72 Himes, Richard H., 217 Holmes, F. Α., 31 Holton, Robert Α., 288 Horwitz, Susan Band, 154 Houze, Jonathan B., 326 Huber, M. H., 31 Jayasinghe, Lalith, 217 Jordon, Mary Ann, 138 Kavanagh, J. J., 31 Keenan, Jeffrey K., 173 Kim, Hyeong-Baik, 288 Kim, Soekchan, 288 Kingston, David G. L, 203 Klein, L. L., 276 Koepp, Alfred, 72 Krauss, Nancy E., 154,326 Kudelka, A. P., 31 Kuduk, Scott D., 262 Lavelle, François, 233,262 Lee, Daesung, 326 Lewis, Norman G., 72 Li, L., 276 Liang, Feng, 288 Liu, Jyanwei H., 288 Lund, M., 189 Manthey, C. L., 162 Marder, R., 189 Maring, C. J., 276 Marquess, Daniel G., 326 Massey, Pamela J., 173 Matiskella, J. D., 124 McGrane, Paul L., 326 Meng, Wei, 326 Mikkilineni, A. B., 124 Monsarrat, B., 98
341 Georg et al.; Taxane Anticancer Agents ACS Symposium Series; American Chemical Society: Washington, DC, 1994.
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342
TAXANE ANTICANCER AGENTS
Mucciaro, Thomas P., 326 Muhlebach, Michel, 326 Millier, R., 189 Murthi, Krishna K., 288 Nadizadeh, Hossain, 288 Natchus, Michael G., 326 Nicolaou, K. C , 302 Ohkuma, Takeshi, 326 Ojima, Iwao, 262 Orr, George Α., 154 Paquette, Leo Α., 313 Park, Haeil, 217 Park, Young Hoon, 262 Pera, Paula, 262 Peschke, Bernd, 326 Plattner, J. J., 276 Potier, P., 189 Rao, Srinivasa, 154 Rawlins, David B., 326 Ringel, Israel, 154 Riou, J. F., 262 Rose, W. C., 124 Royer, L, 98 Sanderink, G. J., 98 Sharma, Α., I l l Sharma, U.S., I l l Shindo, Mitsuru, 288 Shuker, Anthony J., 326 Smith, Chase C , 288 Somoza, Carmen, 288 Stierle, Andrea, 81 Stierle, Donald, 81 Straubinger, R. M., I l l
Strobel, Gary, 81 Suffness, Matthew, 1 Sun, Chung-Ming, 262 Sutton, Jim C , 326 Suzuki, Yukio, 288 Swindell, Charles S., 154 Tang, Suhan, 288 Tao, Chunlin, 288 Taylor, Richard E., 326 Thomas, S. Α., 276 Tomooka, Katsuhiko, 326 Ueda, Y., 124 Valero, V.,31 Vander Velde, David G., 217 Veith, Jean M., 262 Vogel, S. N., 162 Vrignaud, P., 262 Vu, Phong, 288 Vuilhorgne, M., 98 Vyas, D. M., 124 Wahl, Α., 189 Wall, Monroe E., 18 Wani, MansukhC, 18 Wender, Paul Α., 326 Wessjohann, Ludger Α., 326 Whitney, S. Α., 58 Wilson, Leslie, 138 Wong, H., 124 Wright, M., 98 Yeung, C. M., 276 Zhang, Pingsheng, 288 Zucco, Martine, 262
Affiliation Index Abbott Laboratories, 276 Albert Einstein College of Medicine, 154 Bristol-Myers Squibb, 124,162,247 Bryn Mawr College, 154 Centre National de la Recherche Scientifique, 98,189 Florida State University, 288 Grace Cancer Drug Center, 262 Hawaii Biotechnology Group Inc., 81
Montana College of Mineral Science and Technology, 81 Montana State University, 81 National Cancer Institute, 1 Ohio State University, 313 Oread Laboratories, 217 Research Triangle Institute, 18 Rhône-Poulenc Rorer, 98,262,233 Stanford University, 326
Georg et al.; Taxane Anticancer Agents ACS Symposium Series; American Chemical Society: Washington, DC, 1994.
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INDEX
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State University of New YorkBuffalo, 111 State University of New YorkStony Brook, 262 The Hebrew University, 154 The Scripps Research Institute, 302 The University of Texas M. D. Anderson Cancer Center, 31 U.S. Department of Agriculture Forest Service, 58
Uniformed Services University of the Health Sciences, 162 Université di Torino, 262 University of California-San Diego, 302 University of CaUfornia-Santa Barbara, 138 University of Kansas, 217 University of Tennessee, 173 Virginia Polytechnic Institute and State University, 203 Washington State University, 72
Subject Index A Α-ring contracted taxoids from 10-deacetylbaccatin III, synthesis, 193-194 A ring of paclitaxel, synthesis, 304/305 ABC ring of paclitaxel, synthesis, 306-307 20-Acetoxy-4-deacetyl-5-epi-20, 0-secotaxol, 88 Acetoxyoxetane, synthesis, 294-296 13-Acetyl-9(#)-dihydrobaccatin III, chemistry, 276-280 Activity, biological, See Biological activity Af-Acyl paclitaxel analogues, convergent synthetic method, 220-223 Adrenal cell effect intermediate filaments, 178-179 microfilaments, 176-178 microtubules, 179,180r Agronomics, biological production of paclitaxel, 4-5 Aliphatic Af-acyl and Af-oxycarbonyl paclitaxel analogues, convergent synthetic method, 222-223 3'-Alkyl and 3'-alkenyl analogues of docetaxel, 271-273 Anticancer agents, critical objectives in western medicine, 81 Antimitotic activity, docetaxel, 234-235,242-243 Antimitotic drugs, inhibition of microtubule dynamics, 142-143
Antitumor activity 3'-alky 1 and 3'-alkenyl analogues of docetaxel, 273 9(#)-dihydrotaxanes, 276-286 docetaxel, 46 in vivo, cyclohexyl analogues of docetaxel and paclitaxel, 271 paclitaxel, 25i,l 11-120 Apoptotic cell death, induction by paclitaxel, 150 Aromatic N-acyl paclitaxel analogues, convergent synthetic method, 220-222 2-Aroyl-2-benzoyltaxol analogue, synthesis, 211-213 3'-Aryl paclitaxel analogues, biology, 219-220 Assays, chemical production of paclitaxel, 8-9 3 '-(p-Azidobenzamido)taxol competition with paclitaxel for microtubule binding sites, 155,157/ microtubule assembly effect, 155,156/ molecular structure, 155,156/ specific labeling of β-tubulin, 155,158/ 3'-(p-Azidobenzamido)taxol-photolabeled β-tubulin, formic acid digestion products, 155,159-161
Β Β-16 melanoma, activity of paclitaxel, 25,27
Georg et al.; Taxane Anticancer Agents ACS Symposium Series; American Chemical Society: Washington, DC, 1994.
